个人简述:
江苏省高校“青蓝工程” 中青年学术带头人。
科研工作:
承担科研项目:
1. 主持国家自然科学基金项目(20742003,20872181,21172265,21472243)2. 参加国家自然科学基金重大研究计划项目(90713038)3. 参加“重大新药创制”科技重大专项 “十一五”计划项目(2009ZX09501-003)
承担课程:有机合成反应,药物合成反应,化学生物学选论,新药设计与合成
代表性论文:
1.Hai-Qi Zhang, Fei-Hu Gong, Chuan-Gui Li, Chi Zhang ,Yan-Jie Wang, Yun-Gen Xu, Li-Ping Sun*, Design and discovery of 4-anilinoquinazoline-acylamino derivatives as EGFR and VEGFR-2 dual TK inhibitors. Eur. J. Med. Chem. 2016, 109, 371-379.2. Sheng-Wei Yang, Chun-Meng Wang, Kaixiang Tang, Jin-Xin Wang and Li-Ping Sun*, An Efficient Approach to the Total Synthesis of Ammosamide B. Eur. J. Org. Chem. 2016, 5, 1050-1053.3. Meining Wang, Aijun Shen, Chi Zhang, Zilan Song,Jing Ai,Hongchun Liu, Liping Sun,*,Jian Ding, Meiyu Geng,*,and Ao Zhang*, Development of Heat Shock Protein (Hsp90) Inhibitors To Combat Resistance to Tyrosine Kinase Inhibitors through Hsp90−Kinase Interactions, J. Med. Chem. 2016, 59, 5563−5586.4.Ya-Hui Deng, Dan Xu, Ye-Xiang Su, Yi-Juan Cheng, Yan-Li Yang, Xiu-Yun Wang, Juan Zhang, Qi-Dong You* and Li-Ping Sun*,Synthesis and Biological Evaluation of Novel Oxazolo[5,4-d]pyrimidines as Potent VEGFR-2 Inhibitors. Chem. Biodivers. 2015, 12, 528-537.5.Ji-Ping Liu, Ya-Hui Deng, Ling Yang,Yi-Juan Cheng, Lawali Manzo, Li-Ping Sun*and Yu Liu*, CPU-12, a novel synthesized oxazolo[5,4-d]pyrimidine derivative, showed superior anti-angiogenic activity, J. Pharmacol. Sci. 2015, 129, 9-17.
教育背景:
1988年毕业于西北师范大学,1991年获中科院兰州化学物理研究所硕士学位,2004年获香港科技大学博士学位, 2005年1月至2006年1月在新加坡国立大学从事博士后研究。